ibhanile12

Iimveliso

I-Citicolinesodium

Inkcazelo emfutshane:

Igama lemveliso: Citicolinesodium
Inombolo ye-CAS: 33818-15-4
Inombolo yokungena ye-EINECS: 251-689-1
Ifomula yemolekyuli: C14H25N4NaO11P2
Ubunzima bemolekyuli: 510.31


Iinkcukacha zeMveliso

Iithegi zeMveliso

Ifomula yoLwakhiwo

7

Ngokwasemzimbeni
Ukubonakala: umgubo omhlophe wekristale
Ukuxinana.
Indawo yokunyibilika: 259-268°C (dec.)
Indawo yokubilisa.
Refractivity
Indawo yokuflasha.

Idatha yoKhuseleko
Udidi olunobungozi.
Inombolo yoThutho lweeMpahla ezinobungozi.
Ukupakisha udidi.

Isicelo
I-Citicoline ifumaneka njengesongezelelo kumazwe angaphezu kwama-70 phantsi kwamagama ahlukeneyo eemveliso: Cebroton, Ceraxon, Cidilin, Citifar, Cognizin, Difosfocin, Hipercol, NeurAxon, Nicholin, Sinkron, Somazina, Synapsine, Startonyl, Trausan, Xerenoos, njl. kuthathwa njengesongezelelo, i-citicoline i-hydrolyzed kwi-choline kunye ne-cytidine emathunjini.Nje ukuba ezi ziwele umqobo wegazi-ubuchopho zihlaziywa zibe yi-citicoline yi-enzyme yokunciphisa izinga kwi-phosphatidylcholine synthesis, i-CTP-phosphocholine cytidylyltransferase.

I-sodium cytarabine yinto ephilayo ene-chemical formula C14H25N4NaO11P2, i-crystalline powder emhlophe.
Inokubuyisela ngokuthe ngcembe ukusebenza kwamalungu kwi-hemiplegia ebangelwa sistroke, kwaye ingasetyenziselwa ukuphazamiseka kokusebenza kunye nokuphazamiseka kwengqondo okubangelwa kukwenzakala okubukhali kwinkqubo yemithambo-luvo, kunye nesifo se-ischemic cerebrovascular kunye ne-vascular dementia.
Iziphumo ze-Pharmacological
Ikhuthaza i-metabolism ye-cerebral substance kunye nokuphucula ukujikeleza kwe-cerebral ngokunciphisa ukuxhathisa kwi-cerebrovascular kunye nokwandisa ukuhamba kwegazi kwi-cerebral.Kwakhona kwandisa umsebenzi we-brainstem upward reticular activation system, ukuqinisa umsebenzi we-vertebral system kunye nokuphucula ukukhubazeka kwemoto, ngoko kunempembelelo ethile ekukhuthazeni ukubuyiswa komsebenzi wengqondo kunye nokukhuthaza ukuvuswa.Emva kokutofa i-cytophosphorus choline inaliti yesodium, inokungena ngokukhawuleza egazini, kwaye enye yayo inokungena kwizicubu zengqondo ngomqobo wegazi-ingqondo.Inxalenye ye-choline iba ngumnikeli olungileyo we-methylation emzimbeni kwaye ingaba nefuthe le-transmethylation kumachiza amaninzi, kwaye malunga ne-1% ye-choline ikhutshwe kumchamo.


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